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Peds Calc

Safety Information

Acyclovir Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Acyclovir is well tolerated, but renal adjustments and allergy screening are crucial before starting therapy in children.

Clinical Utility: 9/10
1 Clinical Sources
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Absolute contraindication is hypersensitivity to acyclovir or valacyclovir. Relative precautions include renal impairment, dehydration, concomitant nephrotoxic drugs, and underlying neurologic disease that could predispose to neurotoxicity.

Contraindications

Absolute Contraindications (Never Use)

Known serious hypersensitivity to acyclovir, valacyclovir, or formulation components

Recurrent severe rash, angioedema, or anaphylaxis requires selection of an antiviral from a different class.

Relative Contraindications (Use With Caution)

Moderate to severe renal impairment or dehydration

Crystalluria and acute kidney injury are dose-related; adjust dosing, optimise hydration, and monitor renal function.

Concomitant nephrotoxic or neurotoxic medications

Agents such as tacrolimus increase CNS and renal adverse events; observe for neurological symptoms and adjust therapy promptly.

Underlying neurologic disorders or seizures

High-dose IV therapy has precipitated encephalopathy; monitor mental status and consider alternative antivirals if risk is high.

Clinical References

Acyclovir Prescribing Informationโ€ขDailyMed (2024)label