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Safety Information

Ampicillin Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Screen for penicillin allergy, EBV-associated rash risk, and renal function before starting ampicillin.

Clinical Utility: 8/10
2 Clinical Sources
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Absolute contraindications include immediate hypersensitivity to penicillins. Relative cautions include infectious mononucleosis, concomitant allopurinol (rash risk), renal impairment (for IV dosing), and history of severe C. difficile infection.

Contraindications

Absolute Contraindications (Never Use)

Documented anaphylaxis, angioedema, or severe cutaneous adverse reaction to ampicillin or any penicillin-class antibiotic

Documented anaphylaxis, angioedema, or severe cutaneous adverse reaction to ampicillin or any penicillin-class antibiotic

Known hypersensitivity to formulation excipients (e.g., sodium citrate in suspension)

Known hypersensitivity to formulation excipients (e.g., sodium citrate in suspension)

Relative Contraindications (Use With Caution)

Active Epstein-Barr virus infection or acute lymphocytic leukemia—high incidence of morbilliform rash

Active Epstein-Barr virus infection or acute lymphocytic leukemia—high incidence of morbilliform rash

History of Clostridioides difficile infection (monitor for recurrence)

History of Clostridioides difficile infection (monitor for recurrence)

Severe renal impairment or hemodialysis (adjust dosing interval to prevent accumulation)

Severe renal impairment or hemodialysis (adjust dosing interval to prevent accumulation)

Patients with cephalosporin or carbapenem allergy—assess severity before prescribing

Patients with cephalosporin or carbapenem allergy—assess severity before prescribing

Use with allopurinol increases rash risk; counsel families on monitoring

Use with allopurinol increases rash risk; counsel families on monitoring

Pregnancy & Lactation

Ampicillin is widely used for intrapartum prophylaxis; generally compatible with breastfeeding. Monitor infants for diarrhea or candidiasis.

Clinical References

Ampicillin for Injection — DailyMedU.S. National Library of Medicine (2025)Label