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Peds Calc

Safety Information

Esomeprazole Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Esomeprazole shares class contraindications with other proton pump inhibitors—rule out hypersensitivity and reassess long-term therapy hazards before continuing beyond the shortest effective duration.

Clinical Utility: 9/10
2 Clinical Sources
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Absolute contraindications include hypersensitivity to esomeprazole, omeprazole, or substituted benzimidazoles, and concurrent rilpivirine therapy. Relative precautions cover chronic high-dose use, severe hepatic impairment, magnesium depletion, and infections requiring gastric acidity for pathogen control.

Contraindications

Absolute Contraindications (Never Use)

Documented hypersensitivity (anaphylaxis, angioedema, severe cutaneous reaction) to esomeprazole, omeprazole, or other substituted benzimidazole proton pump inhibitors

Documented hypersensitivity (anaphylaxis, angioedema, severe cutaneous reaction) to esomeprazole, omeprazole, or other substituted benzimidazole proton pump inhibitors

Concomitant use with rilpivirine-containing antiretroviral regimens

Concomitant use with rilpivirine-containing antiretroviral regimens

Relative Contraindications (Use With Caution)

Chronic therapy without periodic reassessment—monitor for C. difficile infection and micronutrient deficiencies

Chronic therapy without periodic reassessment—monitor for C. difficile infection and micronutrient deficiencies

History of hypomagnesemia or concurrent diuretic therapy—check magnesium during prolonged use

History of hypomagnesemia or concurrent diuretic therapy—check magnesium during prolonged use

Severe hepatic impairment—reduce maintenance dosing and observe for accumulation

Severe hepatic impairment—reduce maintenance dosing and observe for accumulation

Medications requiring acidic gastric pH for absorption (atazanavir, erlotinib, ketoconazole)—consider alternatives

Medications requiring acidic gastric pH for absorption (atazanavir, erlotinib, ketoconazole)—consider alternatives

High fracture risk or osteoporosis—chronic PPI therapy may reduce calcium absorption

High fracture risk or osteoporosis—chronic PPI therapy may reduce calcium absorption

Clinical References

NASPGHAN Clinical Practice Guideline for Pediatric GERDJ Pediatr Gastroenterol Nutr (2023)guideline