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Peds Calc

Safety Information

Nitazoxanide Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Nitazoxanide treats Giardia, Cryptosporidium, and other protozoal infections. Evaluate hypersensitivity, hepatic function, and immunocompetence before prescribing.

Clinical Utility: 8/10
2 Clinical Sources
Back to Nitazoxanide Overview

Absolute contraindication is hypersensitivity to nitazoxanide or formulation components. Relative contraindications include moderate-to-severe hepatic impairment, severe renal impairment, immunocompromised hosts requiring prolonged therapy, and concomitant drugs that rely on tight hepatic monitoring.

Contraindications

Absolute Contraindications (Never Use)

Hypersensitivity to nitazoxanide, tizoxanide metabolites, or formulation excipients — prior anaphylaxis or severe dermatologic reactions preclude rechallenge.

Hypersensitivity to nitazoxanide, tizoxanide metabolites, or formulation excipients — prior anaphylaxis or severe dermatologic reactions preclude rechallenge.

Relative Contraindications (Use With Caution)

Moderate to severe hepatic impairment or biliary obstruction; metabolism is primarily hepatic, so product labeling recommends closer monitoring of liver enzymes and clinical status.

Moderate to severe hepatic impairment or biliary obstruction; metabolism is primarily hepatic, so product labeling recommends closer monitoring of liver enzymes and clinical status.

Renal impairment with reduced creatinine clearance; metabolites are renally eliminated and accumulation can prolong gastrointestinal adverse effects.

Renal impairment with reduced creatinine clearance; metabolites are renally eliminated and accumulation can prolong gastrointestinal adverse effects.

Immunocompromised hosts (including transplant recipients or advanced HIV) because effectiveness for Cryptosporidium is reduced — coordinate care with infectious diseases specialists and monitor stool studies.

Immunocompromised hosts (including transplant recipients or advanced HIV) because effectiveness for Cryptosporidium is reduced — coordinate care with infectious diseases specialists and monitor stool studies.

Pregnancy and breastfeeding when alternative agents exist; human data remain limited and benefits should clearly outweigh potential fetal or neonatal risk.

Pregnancy and breastfeeding when alternative agents exist; human data remain limited and benefits should clearly outweigh potential fetal or neonatal risk.

Clinical References

CDC Clinical Overview of CryptosporidiosisCenters for Disease Control and Prevention (2024)guideline