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Safety Information

Omeprazole Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Confirm allergy history and assess potential interactions (e.g., clopidogrel).

Clinical Utility: 7/10
2 Clinical Sources
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Absolute: hypersensitivity to omeprazole/PPIs. Relative: risk of CDAD, long‑term use concerns (per clinician), interactions via CYP2C19.

Contraindications

Absolute Contraindications (Never Use)

Documented hypersensitivity (anaphylaxis, angioedema, severe cutaneous reactions) to omeprazole or other substituted benzimidazole PPIs

Documented hypersensitivity (anaphylaxis, angioedema, severe cutaneous reactions) to omeprazole or other substituted benzimidazole PPIs

Concomitant use with rilpivirine-containing antiretroviral products

Concomitant use with rilpivirine-containing antiretroviral products

Relative Contraindications (Use With Caution)

Chronic therapy without periodic reassessment—monitor for C. difficile infection and nutrient malabsorption

Chronic therapy without periodic reassessment—monitor for C. difficile infection and nutrient malabsorption

History of hypomagnesemia, osteoporosis, or long-term diuretic use—check magnesium and bone health during extended courses

History of hypomagnesemia, osteoporosis, or long-term diuretic use—check magnesium and bone health during extended courses

Severe hepatic impairment—reduce maintenance doses and monitor liver function

Severe hepatic impairment—reduce maintenance doses and monitor liver function

Medications requiring acidic gastric pH for absorption (e.g., atazanavir, ketoconazole, erlotinib)—consider alternatives

Medications requiring acidic gastric pH for absorption (e.g., atazanavir, ketoconazole, erlotinib)—consider alternatives

High-dose methotrexate therapy—hold omeprazole around chemotherapy to prevent reduced clearance

High-dose methotrexate therapy—hold omeprazole around chemotherapy to prevent reduced clearance

Clinical References

Omeprazole — FDA DailyMedU.S. National Library of Medicine (2025)Label
Omeprazole — MedlinePlus Drug InformationMedlinePlus / NIH (2025)Database