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Peds Calc

Safety Information

Pantoprazole Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Pantoprazole is often chosen when CYP interactions must be minimized; nonetheless, validate class contraindications and plan for periodic deprescribing discussions.

Clinical Utility: 9/10
2 Clinical Sources
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Absolute contraindications include hypersensitivity to pantoprazole or substituted benzimidazoles, and concomitant use with rilpivirine. Relative issues include chronic therapy without reassessment, hypomagnesemia risk, and infections associated with long-term acid suppression.

Contraindications

Absolute Contraindications (Never Use)

Known hypersensitivity to pantoprazole, other substituted benzimidazole PPIs, or formulation excipients

Known hypersensitivity to pantoprazole, other substituted benzimidazole PPIs, or formulation excipients

History of severe immediate hypersensitivity (anaphylaxis, angioedema) to proton pump inhibitors

History of severe immediate hypersensitivity (anaphylaxis, angioedema) to proton pump inhibitors

Relative Contraindications (Use With Caution)

Concomitant use with rilpivirine-containing antiretroviral regimens (marked loss of virologic efficacy)

Concomitant use with rilpivirine-containing antiretroviral regimens (marked loss of virologic efficacy)

Need for drugs requiring acidic pH for absorption (atazanavir, erlotinib, ketoconazole)—consider alternatives or therapeutic drug monitoring

Need for drugs requiring acidic pH for absorption (atazanavir, erlotinib, ketoconazole)—consider alternatives or therapeutic drug monitoring

Pre-existing hypomagnesemia or long-term diuretic therapy—risk of profound magnesium depletion

Pre-existing hypomagnesemia or long-term diuretic therapy—risk of profound magnesium depletion

High fracture risk or osteoporosis—prolonged PPI use may decrease calcium absorption

High fracture risk or osteoporosis—prolonged PPI use may decrease calcium absorption

History of Clostridioides difficile infection—chronic acid suppression raises recurrence risk

History of Clostridioides difficile infection—chronic acid suppression raises recurrence risk

Clinical References

NASPGHAN Clinical Practice Guideline for Pediatric GERDJ Pediatr Gastroenterol Nutr (2023)guideline