adorable baby smiling with joy

Peds Calc

Safety Information

Terbinafine Contraindications & InteractionsWhen Not to Use & Important Drug Interactions

Most healthy children can take terbinafine safely, but baseline assessment reduces rare hepatotoxicity events.

Clinical Utility: 8/10
2 Clinical Sources
Back to Terbinafine Overview

Absolute: hypersensitivity to terbinafine, chronic or active liver disease. Relative: renal impairment, CYP2D6 substrate co-therapy, psoriasis/lupus flare history, pregnancy.

Contraindications

Absolute Contraindications (Never Use)

History of hypersensitivity to terbinafine or any formulation components

History of hypersensitivity to terbinafine or any formulation components

Active or chronic liver disease with significant hepatic impairment

Active or chronic liver disease with significant hepatic impairment

Relative Contraindications (Use With Caution)

Baseline hepatic dysfunction or elevated transaminases—obtain labs before therapy and monitor every 4–6 weeks during prolonged courses

Baseline hepatic dysfunction or elevated transaminases—obtain labs before therapy and monitor every 4–6 weeks during prolonged courses

Chronic kidney disease with creatinine clearance <50 mL/min

Chronic kidney disease with creatinine clearance <50 mL/min

Concomitant CYP2D6 substrates with narrow therapeutic index (tricyclic antidepressants, some beta-blockers)—consider dose adjustments

Concomitant CYP2D6 substrates with narrow therapeutic index (tricyclic antidepressants, some beta-blockers)—consider dose adjustments

Psoriasis or systemic lupus erythematosus—rare flares reported; monitor skin changes

Psoriasis or systemic lupus erythematosus—rare flares reported; monitor skin changes

Pregnancy or lactation—limited pediatric data; weigh benefits vs risks

Pregnancy or lactation—limited pediatric data; weigh benefits vs risks

Clinical References

Terbinafine Hydrochloride Tablets — DailyMedU.S. National Library of Medicine (2024)Label
TerbinafineStatPearls Publishing (2025)Review